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SYNTHETIC MELANOCYTE STIMULATING HORMONE RELEASE-INHIBITING FACTOR (MIF). III. EFFECT OF L-PROLYL-N-METHYL-D-LEUCYL-GLYCINAMIDE AND MIF ON BIOGENIC AMINE TURNOVER.PUGSLEY TA; LIPPMANN W.1977; ARZNEIMITTEL-FORSCH.; DTSCH.; DA. 1977; VOL. 27; NO 12; PP. 2293-2296; ABS. ALLEM.; BIBL. 37 REF.Article

Comparative pharmacokinetic and pharmacodynamic analysis of phthaloyl glycine derivatives with potential antiepileptic activityOMAR ABU SALACH; SALIM HADAD; ABDULLAH HAJ-YEHIA et al.Pharmaceutical research. 1994, Vol 11, Num 10, pp 1429-1434, issn 0724-8741Article

Novel phenylamino acetamide derivatives as potent and selective κ opioid receptor agonistsCHU, Guo-Hua; MINGHUA GU; DOLLE, Roland E et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 3, pp 645-648, issn 0960-894X, 4 p.Article

Indolyl and dihydroindolyl N-glycinamides as potent and in vivo active NPY5 antagonistsLINGYUN WU; KAI LU; PACKIARAJAN, Mathivanan et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 6, pp 2167-2171, issn 0960-894X, 5 p.Article

Direct Fmoc-Chemistry-Based Solid-Phase Synthesis of Peptidyl ThioestersSHARMA, Indrajeet; CRICH, David.Journal of organic chemistry. 2011, Vol 76, Num 16, pp 6518-6524, issn 0022-3263, 7 p.Article

Convergent synthesis of ribonuclease L-active 2', 5'-oligoadenylate-peptide nucleic acidsZHENGFU WANG; LING CHEN; BAYLY, S. F et al.Bioorganic & medicinal chemistry letters (Print). 2000, Vol 10, Num 12, pp 1357-1360, issn 0960-894XArticle

Bifunctional agents for reperfusion arrhythmias: Novel hybrid vitamin E/class I antiarrhythmicsKOUFAKI, Maria; CALOGEROPOULOU, Theodora; REKKA, Eleni et al.Bioorganic & medicinal chemistry. 2003, Vol 11, Num 23, pp 5209-5219, issn 0968-0896, 11 p.Article

Physicochemical determinants of passive membrane permeability : Role of solute hydrogen-bonding potential and volumeGOODWIN, Jay T; CONRADI, Robert A; HO, Norman F. H et al.Journal of medicinal chemistry (Print). 2001, Vol 44, Num 22, pp 3721-3729, issn 0022-2623Article

Sulfonamido-aryl ethers as bradykinin B1 receptor antagonistsCOLE, Andrew G; METZGER, Axel; RITCHIE, Timothy J et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 1, pp 119-122, issn 0960-894X, 4 p.Article

Design of a radiopharmaceutical for the palliation of painful bone metastases: rhenium-186-labeled bisphosphonate derivativeOGAWA, Kazuma; MUKAI, Takahiro; ARANO, Yasushi et al.Journal of labelled compounds & radiopharmaceuticals. 2004, Vol 47, Num 11, pp 753-761, issn 0362-4803, 9 p.Article

A bivalent ligand (KMN-21) antagonist for μ/κ heterodimeric opioid receptorsSHIJUN ZHANG; YEKKIRALA, Ajay; YE TANG et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 24, pp 6978-6980, issn 0960-894X, 3 p.Article

Discovery of Disubstituted Cyclohexanes as a New Class of CC Chemokine Receptor 2 AntagonistsCHERNEY, Robert J; RUOWEI MO; SOLOMON, Kimberly A et al.Journal of medicinal chemistry (Print). 2008, Vol 51, Num 4, pp 721-724, issn 0022-2623, 4 p.Article

An efficient and versatile synthesis of acylpolyamine spider toxinsNIHEI, Ken-Ichi; KATO, Massuo J; YAMANE, Tetsuo et al.Bioorganic & medicinal chemistry letters (Print). 2002, Vol 12, Num 3, pp 299-302, issn 0960-894XArticle

Novel sulfone-containing di- and trisubstituted cyclohexanes as potent CC chemokine receptor 2 (CCR2) antagonistsCHERNEY, Robert J; RUOWEI MO; DECICCO, Carl P et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 13, pp 3418-3422, issn 0960-894X, 5 p.Article

Identification of Lead Compounds As Antagonists of Protein Bcl-xL with a Diversity-Oriented Multidisciplinary ApproachDI MICCO, Simone; VITALE, Romina; PELLECCHIA, Maurizio et al.Journal of medicinal chemistry (Print). 2009, Vol 52, Num 23, pp 7856-7867, issn 0022-2623, 12 p.Article

Characterization of the binding properties of SIRT2 inhibitors with a N-(3-phenylpropenoyl)-glycine tryptamide backboneKIVIRANTA, Päivi H; SALO, Heikki S; WALLEN, Erik A. A et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 17, pp 8054-8062, issn 0968-0896, 9 p.Article

Discovery of INCB3344, a potent, selective and orally bioavailable antagonist of human and murine CCR2XUE, Chu-Biao; ANLAI WANG; ANAND, Rajan et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 24, pp 7473-7478, issn 0960-894X, 6 p.Article

Design, synthesis and cell growth inhibitory activity of a series of novel aminosubstituted xantheno[1,2-d]imidazoles in breast cancer cellsKOSTAKIS, Ioannis K; POULI, Nicole; MARAKOS, Panagiotis et al.Bioorganic & medicinal chemistry. 2008, Vol 16, Num 6, pp 3445-3455, issn 0968-0896, 11 p.Article

Synthesis and anticonvulsant activity of a class of 2-amino 3-hydroxypropanamide and 2-aminoacetamide derivativesGHIDINI, Eleonora; DELCANALE, Maurizio; BERGAMASCHI, Marco et al.Bioorganic & medicinal chemistry. 2006, Vol 14, Num 10, pp 3263-3274, issn 0968-0896, 12 p.Article

Structure-based discovery of nonpeptidic small organic compounds to block the T cell response to myelin basic proteinKOEHLER, Niklas K. U; YANG, Chao-Yie; LONG, Ya-Qiu et al.Journal of medicinal chemistry (Print). 2004, Vol 47, Num 21, pp 4989-4997, issn 0022-2623, 9 p.Article

Improving potency and selectivity of a new class of non-Zn-chelating MMP-13 inhibitorsHEIM-RIETHER, Alexander; TAYLOR, Steven J; JUNKER, Hans-Dieter et al.Bioorganic & medicinal chemistry letters (Print). 2009, Vol 19, Num 18, pp 5321-5324, issn 0960-894X, 4 p.Article

A new aliphatic amino prodrug system for the delivery of small molecules and proteins utilizing novel PEG derivativesGREENWALD, Richard B; HONG ZHAO; YANG, Karen et al.Journal of medicinal chemistry (Print). 2004, Vol 47, Num 3, pp 726-734, issn 0022-2623, 9 p.Article

Synthesis and biological properties of amino acid amide ligand-based pyridinioalkanoyl thioesters as anti-HIV agentsYONGSHENG SONG; GOEL, Atul; BASRUR, Venkatesha et al.Bioorganic & medicinal chemistry. 2002, Vol 10, Num 5, pp 1263-1273, issn 0968-0896Article

Overcoming hERG activity in the discovery of a series of 4-azetidinyl-1-aryl-cyclohexanes as CCR2 antagonistsXUQING ZHANG; HUFNAGEL, Heather; JOHNSON, Dana et al.Bioorganic & medicinal chemistry letters (Print). 2011, Vol 21, Num 18, pp 5577-5582, issn 0960-894X, 6 p.Article

Synthesis and structure-activity relationships of piperidine-based melanin-concentrating hormone receptor 1 antagonistsWU, Wen-Lian; BURNETT, Duane A; SPRING, Richard et al.Bioorganic & medicinal chemistry letters (Print). 2006, Vol 16, Num 14, pp 3668-3673, issn 0960-894X, 6 p.Article

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